Browsing byAuthorSim, Taebo
Showing results 20 to 49 of 88
| Issue Date | Title | Author(s) |
|---|---|---|
| 2015-07 | Design and Synthesis of New [1,2,3]Triazolo[4,5-d]pyrimidine Derivatives as Potential Antiproliferative Agents | Elkamhawy, Ahmed; Al-Sanea, Mohammad M.; Song, Chiman; Sim, Taebo; Roh, Eun Joo |
| 2011-08 | Design, synthesis, and antiproliferative activity of new 1H-pyrrolo[3,2-c]pyridine derivatives against melanoma cell lines | El-Gamal, Mohammed I.; Jung, Myung-Ho; Lee, Woong San; Sim, Taebo; Yoo, Kyung Ho; Oh, Chang-Hyun |
| 2012-07-01 | Design, synthesis, and antiproliferative activity of new 1H-pyrrolo[3,2-c]pyridine derivatives against melanoma cell lines. Part 2 | Jung, Myung-Ho; El-Gamal, Mohammed I.; Abdel-Maksoud, Mohammed S.; Sim, Taebo; Yoo, Kyung Ho; Oh, Chang-Hyun |
| 2018-12-15 | Design, synthesis, and biological evaluation of novel aminopyrimidinylisoindolines as AXL kinase inhibitors | Choi, Min Jung; Roh, Eun Joo; Hur, Wooyoung; Lee, So Ha; Sim, Taebo; Oh, Chang-Hyun; Lee, Sun-Hwa; Kim, Jong Seung; Yoo, Kyung Ho |
| 2012-08-15 | Development of 'DFG-out' inhibitors of gatekeeper mutant kinases | Choi, Hwan Geun; Zhang, Jianming; Weisberg, Ellen; Griffin, James D.; Sim, Taebo; Gray, Nathanael S. |
| 2019-06 | Development of a Selective CDK7 Covalent Inhibitor Reveals Predominant Cell-Cycle Phenotype | Olson, Calla M.; Liang, Yanke; Leggett, Alan; Park, Woojun D.; Li, Lianbo; Mills, Caitlin E.; Elsarrag, Selma Z.; Ficarro, Scott B.; Zhang, Tinghu; Duester, Robert; Geyer, Matthias; Sim, Taebo; Marto, Jarrod A.; Sorger, Peter K.; Westover, Ken D.; Lin, Charles Y.; Kwiatkowski, Nicholas; Gray, Nathanael S. |
| 2016-08 | Development of Chemical Probes for Investigation of Salt-Inducible Kinase Function in Vivo | Sundberg, Thomas B.; Liang, Yanke; Wu, Huixian; Choi, Hwan Geun; Kim, Nam Doo; Sim, Taebo; Johannessen, Liv; Petrone, Adam; Khor, Bernard; Graham, Daniel B.; Latorre, Isabel J.; Phillips, Andrew J.; Schreiber, Stuart L.; Perez, Jose; Shamji, Alykhan F.; Gray, Nathanael S.; Xavier, Ramnik J. |
| 2014-11-11 | Development of covalent inhibitors that can overcome resistance to first-generation FGFR kinase inhibitors | Tan, Li; Wang, Jun; Tanizaki, Junko; Huang, Zhifeng; Aref, Amir R.; Rusan, Maria; Zhu, Su-Jie; Zhang, Yiyun; Ercan, Dalia; Liao, Rachel G.; Capelletti, Marzia; Zhou, Wenjun; Hur, Wooyoung; Kim, NamDoo; Sim, Taebo; Gaudet, Suzanne; Barbie, David A.; Yeh, Jing-Ruey Joanna; Yun, Cai-Hong; Hammerman, Peter S.; Mohammadi, Moosa; Jaenne, Pasi A.; Gray, Nathanael S. |
| 2018-06 | Development of Highly Potent and Selective Steroidal Inhibitors and Degraders of CDK8 | Hatcher, John M.; Wang, Eric S.; Johannessen, Liv; Kwiatkowski, Nicholas; Sim, Taebo; Gray, Nathanael S. |
| 2010-03-01 | Discovery and initial SAR of pyrimidin-4-yl-1H-imidazole derivatives with antiproliferative activity against melanoma cell lines | Lee, Junghun; Kim, Hwan; Yu, Hana; Chung, Jae Yoon; Oh, Chang-Hyun; Yoo, Kyung Ho; Sim, Taebo; Hah, Jung-Mi |
| 2016-01-02 | Discovery of a broad spectrum antiproliferative agent with selectivity for DDR1 kinase: cell line-based assay, kinase panel, molecular docking, and toxicity studies | Elkamhawy, Ahmed; Park, Jung-eun; Cho, Nam-Chul; Sim, Taebo; Pae, Ae Nim; Roh, Eun Joo |
| 2016-05 | Discovery of a Highly Potent and Selective Indenoindolone Type 1 Pan-FLT3 Inhibitor | Hatcher, John M.; Weisberg, Ellen; Sim, Taebo; Stone, Richard M.; Liu, Suiyang; Griffin, James D.; Gray, Nathanael S. |
| 2015-08-16 | Discovery of a potent, selective inhibitor of RET kinase including the V804L/V804M gatekeeper mutants | Yoon, Hojong; Kwak, Yeonui; Sim, Taebo; Kim, Nam Doo; Cho, Kyung Seon; Choi, Seunghye |
| 2016-10 | Discovery of a Series of 5,11-Dihydro-6H-benzo[e]pyrimido[5,4-b][1,4]diazepin-6-ones as Selective PI3K-delta/gamma Inhibitors | Ferguson, Fleur M.; Ni, Jing; Zhang, Tinghu; Tesar, Bethany; Sim, Taebo; Kim, Nam Doo; Deng, Xianming; Brown, Jennifer R.; Zhao, Jean J.; Gray, Nathanael S. |
| 2019-06 | Discovery of Covalent CDK14 Inhibitors with Pan-TAIRE Family Specificity | Ferguson, Fleur M.; Doctor, Zainab M.; Ficarro, Scott B.; Browne, Christopher M.; Marto, Jarrod A.; Johnson, Jared L.; Yaron, Tomer M.; Cantley, Lewis C.; Kim, Nam Doo; Sim, Taebo; Berberich, Matthew J.; Kalocsay, Marian; Sorger, Peter K.; Gray, Nathanael S. |
| 2015-12-10 | Discovery of Inhibitors That Overcome the G1202R Anaplastic Lymphoma Kinase Resistance Mutation | Hatcher, John M.; Bahcall, Magda; Choi, Hwan Geun; Gao, Yang; Sim, Taebo; George, Rani; Jaenne, Pasi A.; Gray, Nathanael S. |
| 2012-01-27 | Discovery of Potent and Selective Covalent Inhibitors of JNK | Zhang, Tinghu; Inesta-Vaquera, Francisco; Niepel, Mario; Zhang, Jianming; Ficarro, Scott B.; Machleidt, Thomas; Xie, Ting; Marto, Jarrod A.; Kim, NamDoo; Sim, Taebo; Laughlin, John D.; Park, Hajeung; LoGrasso, Philip V.; Patricelli, Matt; Nomanbhoy, Tyzoon K.; Sorger, Peter K.; Alessi, Dario R.; Gray, Nathanael S. |
| 2015-01-08 | Discovery of Type II Inhibitors of TGF beta-Activated Kinase 1 (TAK1) and Mitogen-Activated Protein Kinase Kinase Kinase Kinase 2 (MAP4K2) | Tan, Li; Nomanbhoy, Tyzoon; Gurbani, Deepak; Patricelli, Matthew; Hunter, John; Geng, Jiefei; Herhaus, Lina; Zhang, Jianming; Pauls, Eduardo; Ham, Youngjin; Choi, Hwan Geun; Xie, Ting; Deng, Xianming; Buhrlage, Sara J.; Sim, Taebo; Cohen, Philip; Sapkota, Gopal; Westover, Kenneth D.; Gray, Nathanael S. |
| 2010-10-14 | Expanding the Diversity of Allosteric Ber-Abl Inhibitors | Deng, Xianming; Okram, Barun; Ding, Qiang; Zhang, Jianming; Choi, Yongmun; Adrian, Francisco J.; Wojciechowski, Amy; Zhang, Guobao; Che, Jianwei; Bursulaya, Badry; Cowan-Jacob, Sandra W.; Rummel, Gabriele; Sim, Taebo; Gray, Nathanael S. |
| 2018-09-27 | First SAR Study for Overriding NRAS Mutant Driven Acute Myeloid Leukemia | Cho, Hanna; Shin, Injae; Ju, Eunhye; Choi, Seunghye; Hur, Wooyoung; Kim, Haelee; Hong, Eunmi; Kim, Nam Doo; Choi, Hwan Geun; Gray, Nathanael S.; Sim, Taebo |
| 2017-02-23 | Highly stereoselective synthesis of mupirocin H | Sengupta, Sandip; Kim, Hak Joong; Cho, Kyung Seon; Song, Woon Young; Sim, Taebo |
| 2019-01-01 | Identification of 1H-pyrazolo[3,4-b]pyridine derivatives as potent ALK-L1196M inhibitors | Nam, Yunju; Hwang, Dongkeun; Kim, Namdoo; Seo, Hong-Seog; Selim, Khalid B.; Sim, Taebo |
| 2017-01-05 | Identification of a novel 5-amino-3-(5-cyclopropylisoxazol-3-yl)-1-isopropyl-1H-pyrazole-4-carboxa mide as a specific RET kinase inhibitor | Yoon, Hojong; Shin, Injae; Nam, Yunju; Kim, Nam Doo; Lee, Kyung-Bok; Sim, Taebo |
| 2019-10-24 | Identification of a Unique Resorcylic Acid Lactone Derivative That Targets Both Lymphangiogenesis and Angiogenesis | Han, Youngsun; Sengupta, Sandip; Lee, Byung Joo; Cho, Hanna; Kim, Jiknyeo; Choi, Hwan Geun; Dash, Uttam; Kim, Jin Hyoung; Kim, Nam Doo; Kim, Jeong Hun; Sim, Taebo |
| 2017-01-01 | Identification of Existing Drugs That Effectively Target NTRK1 and ROS1 Rearrangements in Lung Cancer | Chong, Curtis R.; Bahcall, Magda; Capelletti, Marzia; Kosaka, Takayuki; Ercan, Dalia; Sim, Taebo; Sholl, Lynette M.; Nishino, Mizuki; Johnson, Bruce E.; Gray, Nathanael S.; Janne, Pasi A. |
| 2013-07-26 | Identification of methyl violet 2B as a novel blocker of focal adhesion kinase signaling pathway in cancer cells | Kim, Hwan; Kim, Nam Doo; Lee, Jiyeon; Han, Gyoonhee; Sim, Taebo |
| 2019-09-26 | Identification of Novel Resorcinol Amide Derivatives as Potent and Specific Pyruvate Dehydrogenase Kinase (PDHK) Inhibitors | Cho, Hanna; Shin, Injae; Cho, Kyungseon; Yoon, Hojong; Yoo, Eun Kyung; Kim, Mi-Jin; Park, Sungmi; Lee, In-Kyu; Kim, Nam Doo; Sim, Taebo |
| 2015-05-14 | Identification of Novel ROS Inducers: Quinone Derivatives Tethered to Long Hydrocarbon Chains | Hong, Yeonsun; Sengupta, Sandip; Hur, Wooyoung; Sim, Taebo |
| 2015-05-14 | Identification of novel therapeutic targets in acute leukemias with NRAS mutations using a pharmacologic approach | Nonami, Atsushi; Sattler, Martin; Weisberg, Ellen; Liu, Qingsong; Zhang, Jianming; Patricelli, Matthew P.; Christie, Amanda L.; Saur, Amy M.; Kohl, Nancy E.; Kung, Andrew L.; Yoon, Hojong; Sim, Taebo; Gray, Nathanael S.; Griffin, James D. |
| 2022-04 | Identification of Pyridinyltriazine Derivatives as Potent panFGFR Inhibitors against Gatekeeper Mutants for Overcoming Drug Resistance | Ryu, SeongShick; Nam, Yunju; Kim, Namkyoung; Shin, Injae; Jeon, Eunhye; Kim, Younghoon; Kim, Nam Doo; Sim, Taebo |
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