Showing results 1 to 13 of 13
Issue Date | Title | Author(s) |
---|---|---|
2016-09 | A Divergent Approach for the Synthesis of D- and L-4 '-Ethynyl Dioxolane Nucleosides with Potent Anti-HIV Activity | Singh, Sarbjit; Gajulapati, Veeraswamy; Kim, Minkyoung; Goo, Ja-Il; Lee, Jae Kyun; Lee, Kyeong; Lee, Chong-Kyo; Jeong, Lak Shin; Choi, Yongseok |
2020-12-10 | Development of a Polo-like Kinase-1 Polo-Box Domain Inhibitor as a Tumor Growth Suppressor in Mice Models | Gunasekaran, Pethaiah; Yim, Min Su; Ahn, Mija; Soung, Nak-Kyun; Park, Jung-Eun; Kim, Jaehi; Bang, Geul; Shin, Sang Chul; Choi, Joonhyeok; Kim, Minkyoung; Kim, Hak Nam; Lee, Young-Ho; Chung, Young-Ho; Lee, Kyeong; Kim, Eunice EunKyeong; Jeon, Young-Ho; Kim, Min Ju; Lee, Kyeong-Ryoon; Kim, Bo-Yeon; Lee, Kyung S.; Ryu, Eun Kyoung; Bang, Jeong Kyu |
2021-09 | Development of New Meridianin/Leucettine-Derived Hybrid Small Molecules as Nanomolar Multi-Kinase Inhibitors with Antitumor Activity | Elsherbeny, Mohamed H.; Elkamhawy, Ahmed; Nada, Hossam; Abdellattif, Magda H.; Lee, Kyeong; Roh, Eun Joo |
2021-11 | Discovery of 3,4-dichloro-N-(1H-indol-5-yl)benzamide: A highly potent, selective, and competitive hMAO-B inhibitor with high BBB permeability and action | Elkamhawy, Ahmed; Kim, Hyeon Jeong; Elsherbeny, Mohamed H.; Paik, Sora; Park, Jong-Hyun; Gotina, Lizaveta; Abdellattif, Magda H.; Gouda, Noha A.; Cho, Jungsook; Lee, Kyeong; Pae, Ae Nim; Park, Ki Duk; Roh, Eun Joo |
2020-01 | Discovery of N-(1-(3-fluorobenzoyl)-1H-indol-5-yl)pyrazine-2-carboxamide: a novel, selective, and competitive indole-based lead inhibitor for human monoamine oxidase B | Elkamhawy, Ahmed; Paik, Sora; Kim, Hyeon Jeong; Park, Jong-Hyun; Londhe, Ashwini M.; Lee, Kyeong; Pae, Ae Nim; Park, Ki Duk; Roh, Eun Joo |
2022-09 | Identification of Novel Aryl Carboxamide Derivatives as Death-Associated Protein Kinase 1 (DAPK1) Inhibitors with Anti-Proliferative Activities: Design, Synthesis, In Vitro, and In Silico Biological Studies | Elkamhawy, Ahmed; Paik, Sora; Ali, Eslam M. H.; Hassan, Ahmed H. E.; Kang, So Jin; Lee, Kyeong; Roh, Eun Joo |
2022-03 | Identification of novel discoidin domain receptor 1 (DDR1) inhibitors using E-pharmacophore modeling, structure-based virtual screening, molecular dynamics simulation and MM-GBSA approaches | Nada, Hossam; Lee, Kyeong; Gotina, Lizaveta; Pae, Ae Nim; Elkamhawy, Ahmed |
2018-11-05 | Iodine-Promoted One-pot Synthesis of Highly Substituted 4-Aminopyrroles and Bis-4-aminopyrrole from Aryl Methyl Ketones, Arylamines, and Enamines | Jalani, Hitesh B.; Mali, Jyotirling R.; Park, Hyejun; Lee, Jae Kyun; Lee, Kiho; Lee, Kyeong; Choi, Yongseok |
2010-10-01 | LW6, a novel HIF-1 inhibitor, promotes proteasomal degradation of HIF-1 alpha via upregulation of VHL in a colon cancer cell line | Lee, Kyeong; Kang, Jung Eun; Park, Song-Kyu; Jin, Yinglan; Chung, Kyung-Sook; Kim, Hwan-Mook; Lee, Kiho; Kang, Moo Rim; Lee, Myung Kyu; Song, Kyung Bin; Yang, Eun-Gyeong; Lee, Jung-Jun; Won, Misun |
2021-10 | Melatonin Analogues Potently Inhibit MAO-B and Protect PC12 Cells against Oxidative Stress | Elkamhawy, Ahmed; Woo, Jiyu; Gouda, Noha A.; Kim, Jushin; Nada, Hossam; Roh, Eun Joo; Park, Ki Duk; Cho, Jungsook; Lee, Kyeong |
2022-09 | Metal/catalyst-free sequential C-N bond forming cascades at room temperature: environment-friendly one-pot synthesis of 5-aminoimidazoles from aryl glyoxals, anilines, and amidines | Jalani, Hitesh B.; Sivaraman, Aneesh; Min, Kyoung Ho; Lee, Hwa Young; Oh, Na Kyoung; Kang, Hyeseul; Keum, Gyochang; Choi, Yongseok; Lee, Kyeong |
2021-09 | Scaffold Repurposing of In-House Small Molecule Candidates Leads to Discovery of First-in-Class CDK-1/HER-2 Dual Inhibitors: In Vitro and In Silico Screening | Elkamhawy, Ahmed; Ammar, Usama M.; Paik, Sora; Abdellattif, Magda H.; Elsherbeny, Mohamed H.; Lee, Kyeong; Roh, Eun Joo |
2020-07 | Sulfonamide-based 4-anilinoquinoline derivatives as novel dual Aurora kinase (AURKA/B) inhibitors: Synthesis, biological evaluation and in silico insights | Al-Sanea, Mohammad M.; Elkamhawy, Ahmed; Paik, Sora; Lee, Kyeong; El Kerdawy, Ahmed M.; Abbas, Bukhari Syed Nasir; Roh, Eun Joo; Eldehna, Wagdy M.; Elshemy, Heba A. H.; Bakr, Rania B.; Farahat, Ibrahim Ali; Alzarea, Abdulaziz, I; Alzarea, Sami, I; Alharbi, Khalid S.; Abdelgawad, Mohamed A. |