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<dcvalue element="contributor" qualifier="author">Ammar,&#x20;Usama&#x20;M.</dcvalue>
<dcvalue element="contributor" qualifier="author">Abdel-Maksoud,&#x20;Mohammed&#x20;S.</dcvalue>
<dcvalue element="contributor" qualifier="author">Ali,&#x20;Eslam&#x20;M.&#x20;H.</dcvalue>
<dcvalue element="contributor" qualifier="author">Mersal,&#x20;Karim,&#x20;I</dcvalue>
<dcvalue element="contributor" qualifier="author">Yoo,&#x20;Kyung&#x20;Ho</dcvalue>
<dcvalue element="contributor" qualifier="author">Oh,&#x20;Chang-Hyun</dcvalue>
<dcvalue element="date" qualifier="accessioned">2024-01-19T17:04:00Z</dcvalue>
<dcvalue element="date" qualifier="available">2024-01-19T17:04:00Z</dcvalue>
<dcvalue element="date" qualifier="created">2022-01-10</dcvalue>
<dcvalue element="date" qualifier="issued">2020-07</dcvalue>
<dcvalue element="identifier" qualifier="issn">0045-2068</dcvalue>
<dcvalue element="identifier" qualifier="uri">https:&#x2F;&#x2F;pubs.kist.re.kr&#x2F;handle&#x2F;201004&#x2F;118430</dcvalue>
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<dcvalue element="publisher" qualifier="none">ACADEMIC&#x20;PRESS&#x20;INC&#x20;ELSEVIER&#x20;SCIENCE</dcvalue>
<dcvalue element="subject" qualifier="none">BIOLOGICAL&#x20;EVALUATION</dcvalue>
<dcvalue element="subject" qualifier="none">MALIGNANT-MELANOMA</dcvalue>
<dcvalue element="subject" qualifier="none">BRAF</dcvalue>
<dcvalue element="subject" qualifier="none">MUTATIONS</dcvalue>
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<dcvalue element="subject" qualifier="none">KINASE</dcvalue>
<dcvalue element="title" qualifier="none">Structural&#x20;optimization&#x20;of&#x20;imidazothiazole&#x20;derivatives&#x20;affords&#x20;a&#x20;new&#x20;promising&#x20;series&#x20;as&#x20;B-Raf&#x20;V600E&#x20;inhibitors;&#x20;synthesis,&#x20;in&#x20;vitro&#x20;assay&#x20;and&#x20;in&#x20;silico&#x20;screening</dcvalue>
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<dcvalue element="identifier" qualifier="doi">10.1016&#x2F;j.bioorg.2020.103967</dcvalue>
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<dcvalue element="identifier" qualifier="bibliographicCitation">BIOORGANIC&#x20;CHEMISTRY,&#x20;v.100</dcvalue>
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<dcvalue element="description" qualifier="journalRegisteredClass">scopus</dcvalue>
<dcvalue element="identifier" qualifier="wosid">000540960000003</dcvalue>
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<dcvalue element="relation" qualifier="journalWebOfScienceCategory">Chemistry,&#x20;Organic</dcvalue>
<dcvalue element="relation" qualifier="journalResearchArea">Biochemistry&#x20;&amp;&#x20;Molecular&#x20;Biology</dcvalue>
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<dcvalue element="subject" qualifier="keywordPlus">BIOLOGICAL&#x20;EVALUATION</dcvalue>
<dcvalue element="subject" qualifier="keywordPlus">MALIGNANT-MELANOMA</dcvalue>
<dcvalue element="subject" qualifier="keywordPlus">BRAF</dcvalue>
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<dcvalue element="subject" qualifier="keywordPlus">VEMURAFENIB</dcvalue>
<dcvalue element="subject" qualifier="keywordPlus">GROWTH</dcvalue>
<dcvalue element="subject" qualifier="keywordPlus">AGENTS</dcvalue>
<dcvalue element="subject" qualifier="keywordPlus">KINASE</dcvalue>
<dcvalue element="subject" qualifier="keywordAuthor">anti&#x20;cancer</dcvalue>
<dcvalue element="subject" qualifier="keywordAuthor">B-Raf&#x20;V600E</dcvalue>
<dcvalue element="subject" qualifier="keywordAuthor">Imidazo[2,1-b]thiazole</dcvalue>
<dcvalue element="subject" qualifier="keywordAuthor">In&#x20;silico&#x20;screening</dcvalue>
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