Kim, SN Lee, JY Kim, HJ Shin, CG Park, H Lee, YS 2024-01-21T13:38:02Z 2024-01-21T13:38:02Z 2021-09-05 2000-08 0960-894X https://pubs.kist.re.kr/handle/201004/141163 Caffeoylglucosides, which have a glucose ring as a central linker, were synthesized from methyl D-glucosides, and their anti-HIV-1 activities were tested. Among them, four dicaffeoylglucosides (IC50 = 29.1-35.1 mu M), 6a, 6b, 9b and 10b, showed HIV-1 integrase inhibitory activity as potent as L-chicoric acid. (C) 2000 Elsevier Science Ltd. All rights reserved. English PERGAMON-ELSEVIER SCIENCE LTD Synthesis and HIV-1 integrase inhibitory activities of caffeoylglucosides Article 10.1016/S0960-894X(00)00355-3 1 BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, v.10, no.16, pp.1879 - 1882 BIOORGANIC & MEDICINAL CHEMISTRY LETTERS 10 16 1879 1882 N scie scopus 000088837600025 2-s2.0-0034698891 Chemistry, Medicinal Chemistry, Organic Pharmacology & Pharmacy Chemistry Article IMMUNODEFICIENCY-VIRUS TYPE-1 DICAFFEOYLTARTARIC ACIDS POTENT INHIBITORS REPLICATION ANALOGS AIDS