Showing results 4 to 9 of 9
Issue Date | Title | Author(s) |
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2019-06 | Leveraging Compound Promiscuity to Identify Targetable Cysteines within the Kinome | Rao, Suman; Gurbani, Deepak; Du, Guangyan; Everley, Robert A.; Browne, Christopher M.; Chaikuad, Apirat; Tan, Li; Schroeder, Martin; Gondi, Sudershan; Ficarro, Scott B.; Sim, Taebo; Kim, Nam Doo; Berberich, Matthew J.; Knapp, Stefan; Marto, Jarrod A.; Westover, Kenneth D.; Sorger, Peter K.; Gray, Nathanael S. |
2014-12 | Pharmacological targeting of the pseudokinase Her3 | Xie, Ting; Lim, Sang Min; Westover, Kenneth D.; Dodge, Michael E.; Ercan, Dalia; Ficarro, Scott B.; Udayakumar, Durga; Gurbani, Deepak; Tae, Hyun Seop; Riddle, Steven M.; Sim, Taebo; Marto, Jarrod A.; Jaenne, Pasi A.; Crews, Craig M.; Gray, Nathanael S. |
2013-03 | Structure and Ubiquitination-Dependent Activation of TANK-Binding Kinase 1 | Tu, Daqi; Zhu, Zehua; Zhou, Alicia Y.; Yun, Cai-hong; Lee, Kyung-Eun; Toms, Angela V.; Li, Yiqun; Dunn, Gavin P.; Chan, Edmond; Tran Thai; Yang, Shenghong; Ficarro, Scott B.; Marto, Jarrod A.; Jeon, Hyesung; Hahn, William C.; Barbie, David A.; Eck, Michael J. |
2019-08 | Synthesis and structure activity relationships of a series of 4-amino-1H-pyrazoles as covalent inhibitors of CDK14 | Ferguson, Fleur M.; Doctor, Zainab M.; Ficarro, Scott B.; Marto, Jarrod A.; Kim, Nam Doo; Sim, Taebo; Gray, Nathanael S. |
2014-07-30 | Targeting transcription regulation in cancer with a covalent CDK7 inhibitor | Kwiatkowski, Nicholas; Zhang, Tinghu; Rahl, Peter B.; Abraham, Brian J.; Reddy, Jessica; Ficarro, Scott B.; Dastur, Anahita; Amzallag, Arnaud; Ramaswamy, Sridhar; Tesar, Bethany; Jenkins, Catherine E.; Hannett, Nancy M.; McMillin, Douglas; Sanda, Takaomi; Sim, Taebo; Kim, Nam Doo; Look, Thomas; Mitsiades, Constantine S.; Weng, Andrew P.; Brown, Jennifer R.; Benes, Cyril H.; Marto, Jarrod A.; Young, Richard A.; Gray, Nathanael S. |
2014-01-03 | Therapeutic Targeting of Oncogenic K-Ras by a Covalent Catalytic Site Inhibitor | Lim, Sang Min; Westover, Kenneth D.; Ficarro, Scott B.; Harrison, Rane A.; Choi, Hwan Geun; Pacold, Michael E.; Carrasco, Martin; Hunter, John; Kim, Nam Doo; Xie, Ting; Sim, Taebo; Jaenne, Pasi A.; Meyerson, Matthew; Marto, Jarrod A.; Engen, John R.; Gray, Nathanael S. |