Browsing byAuthorRoh, Eun Joo
Showing results 30 to 59 of 66
| Issue Date | Title | Author(s) |
|---|---|---|
| 2022-09 | Identification of Novel Aryl Carboxamide Derivatives as Death-Associated Protein Kinase 1 (DAPK1) Inhibitors with Anti-Proliferative Activities: Design, Synthesis, In Vitro, and In Silico Biological Studies | Elkamhawy, Ahmed; Paik, Sora; Ali, Eslam M. H.; Hassan, Ahmed H. E.; Kang, So Jin; Lee, Kyeong; Roh, Eun Joo |
| 2024-01 | Integrating computational methods guided the discovery of phytochemicals as potential Pin1 inhibitors for cancer: pharmacophore modeling, molecular docking, MM-GBSA calculations and molecular dynamics studies | Alzain, Abdulrahim A.; Elbadwi, Fatima A.; Shoaib, Tagyedeen H.; Sherif, Asmaa E.; Osman, Wadah; Ashour, Ahmed; Mohamed, Gamal A.; Ibrahim, Sabrin R. M.; Roh, Eun Joo; Hassan, Ahmed H. E. |
| 2007-02-01 | Lead discovery and optimization of T-type calcium channel blockers | Park, Jung Hwan; Choi, Jin Kyu; Lee, Eunjung; Lee, Jae Kyun; Rhim, Hyewhon; Seo, Seon Hee; Kim, Yoonjee; Doddareddy, Munikumar Reddy; Pae, Ae Nim; Kang, Jahyo; Roh, Eun Joo |
| 2021-10 | Melatonin Analogues Potently Inhibit MAO-B and Protect PC12 Cells against Oxidative Stress | Elkamhawy, Ahmed; Woo, Jiyu; Gouda, Noha A.; Kim, Jushin; Nada, Hossam; Roh, Eun Joo; Park, Ki Duk; Cho, Jungsook; Lee, Kyeong |
| 2013-11 | MONNA, a Potent and Selective Blocker for Transmembrane Protein with Unknown Function 16/Anoctamin-1 | Oh, Soo-Jin; Hwang, Seok Jin; Jung, Jonghoon; Yu, Kuai; Kim, Jeongyeon; Choi, Jung Yoon; Hartzell, H. Criss; Roh, Eun Joo; Lee, C. Justin |
| 2017-12-01 | Novel LCK/FMS inhibitors based on phenoxypyrimidine scaffold as potential treatment for inflammatory disorders | Farag, Ahmed Karam; Elkamhawy, Ahmed; Londhe, Ashwini M.; Lee, Kyung-Tae; Pae, Ae Nim; Roh, Eun Joo |
| 2023-09 | Novel potent blockers for TWIK-1/TREK-1 heterodimers as potential antidepressants | Lee, Elliot H.; Park, Jung-eun; Gotina, Lizaveta; Han, Young-Eun; Viswanath, Ambily Nath Indu; Yoo, Seonguk; Moon, Bongjin; Hwang, Jin-Young; Park, Woo Kyu; Cho, Yoonjeong; Song, Chiman; Min, Sun-Joon; Hwang, Eun Mi; Lee, Hyunbeom; Pae, Ae Nim; Roh, Eun Joo; Oh, Soo-Jin |
| 2014-09-12 | Novel quinazoline-urea analogues as modulators for A beta-induced mitochondrial dysfunction: Design, synthesis, and molecular docking study | Elkamhawy, Ahmed; Lee, Jiyoun; Park, Beoung-Geon; Park, Insun; Pae, Ae Nim; Roh, Eun Joo |
| 2018-11 | Novel Rhodanine Derivative, 5-[4-(4-Fluorophenoxy)phenyl]methylene-3-{4-[3-(4-methylpiperazin-1-yl)p ropoxy]phenyl}-2-thioxo-4-thiazolidinone dihydrochloride, Induces Apoptosis via Mitochondria Dysfunction and Endoplasmic Reticulum Stress in Human Colon Cancer Cells | Jung, Hye-Uk; Lee, Jeong-Hun; Chung, Kyung-Sook; Hong, Joo Young; Choi, Jung-Hye; Kim, Soo-Dong; Roh, Eun Joo; Shin, Kye Jung; Lee, Kyung-Tae |
| 2023-05 | Novel topoisomerase II/EGFR dual inhibitors: design, synthesis and docking studies of naphtho[2',3':4,5]thiazolo[3,2-a]pyrimidine hybrids as potential anticancer agents with apoptosis inducing activity | Mourad, Mai A. E.; Elmaaty, Ayman Abo; Zaki, Islam; Mourad, Ahmed A. E.; Hofni, Amal; Khodir, Ahmed E.; Aboubakr, Esam M.; Elkamhawy, Ahmed; Roh, Eun Joo; Al-Karmalawy, Ahmed A. |
| 2019-11 | Optimization study towards more potent thiazolidine-2,4-dione IKK-beta modulator: Synthesis, biological evaluation and in silico docking simulation | Elkamhawy, Ahmed; Kim, Nam Youn; Hassan, Ahmed H. E.; Park, Jung-eun; Yang, Jeong-Eun; Elsherbeny, Mohamed H.; Paik, Sora; Oh, Kwang-Seok; Lee, Byung Ho; Lee, Mi Young; Shin, Kye Jung; Pae, Ae Nim; Lee, Kyung-Tae; Roh, Eun Joo |
| 2008-09-20 | Organic Solvents Containing Zwitterion as Electrolyte for Li Ion Cells | Krishnan, Jegatha Nambi; Kim, Hyung Sun; Lee, Jae Kyun; Cho, Byung-Won; Roh, Eun Joo; Lee, Sang-Gi |
| 2007-07-12 | P2Y(1) antagonists: Combining receptor-based modeling and QSAR for a quantitative prediction of the biological activity based on consensus scoring | Costanzi, Stefano; Tikhonova, Irina G.; Ohno, Michihiro; Roh, Eun Joo; Joshi, Bhalchandra V.; Colson, Anny-Odile; Houston, Dayle; Maddileti, Savitri; Harden, T. Kendall; Jacobson, Kenneth A. |
| 2018-09-05 | Pyrazinyl ureas revisited: 1-(3-(Benzyloxy)pyrazin-2-yl)-3-(3,4-dichlorophenyl)urea, a new blocker of A beta-induced mPTP opening for Alzheimer's disease | Elkamhawy, Ahmed; Park, Jung-eun; Hassan, Ahmed H. E.; Pae, Ae Nim; Lee, Jiyoun; Paik, Sora; Park, Beoung-Geon; Roh, Eun Joo |
| 2018-05-10 | Repositioning of the antipsychotic trifluoperazine: Synthesis, biological evaluation and in silico study of trifluoperazine analogs as anti-glioblastoma agents | Kang, Seokmin; Lee, Jung Moo; Jeon, Borami; Elkamhawy, Ahmed; Paik, Sora; Hong, Jinpyo; Oh, Soo-Jin; Paek, Sun Ha; Lee, C. Justin; Hassan, Ahmed H. E.; Kang, Sang Soo; Roh, Eun Joo |
| 2020-01-01 | Reprofiling of pyrimidine-based DAPK1/CSF1R dual inhibitors: identification of 2,5-diamino-4-pyrimidinol derivatives as novel potential anticancer lead compounds | Farag, Ahmed K.; Hassan, Ahmed H. E.; Ahn, Byung Sun; Park, Ki Duk; Roh, Eun Joo |
| 2021-09 | Scaffold Repurposing of In-House Small Molecule Candidates Leads to Discovery of First-in-Class CDK-1/HER-2 Dual Inhibitors: In Vitro and In Silico Screening | Elkamhawy, Ahmed; Ammar, Usama M.; Paik, Sora; Abdellattif, Magda H.; Elsherbeny, Mohamed H.; Lee, Kyeong; Roh, Eun Joo |
| 2012-08-15 | Small molecules that protect against beta-amyloid-induced cytotoxicity by inhibiting aggregation of beta-amyloid | Lee, Yun Suk; Kim, Hye Yun; Kim, YoungSoo; Seo, Jae Hong; Roh, Eun Joo; Han, Hogyu; Shin, Kye Jung |
| 2013-02-06 | Stereoselective synthesis of (-)-8-epi-swainsonine starting with a chiral aziridine | Lee, Baeck Kyoung; Choi, Hwan Geun; Roh, Eun Joo; Lee, Won Koo; Sim, Taebo |
| 2008-10-15 | Structure-activity relationships of 1,4-dihydropyridines that act as enhancers of the vanilloid receptor 1 (TRPV1) | Roh, Eun Joo; Keller, Jason M.; Olah, Zoltan; Iadarola, Michael J.; Jacobson, Kenneth A. |
| 2014-08-01 | Structure-based optimization and biological evaluation of trisubstituted pyrazole as a core structure of potent ROS1 kinase inhibitors | Park, Byung Sun; Al-Sanea, Mohammad M.; Abdelazem, Ahmed Z.; Park, Hye Mi; Roh, Eun Joo; Park, Hyun-Mee; Yoo, Kyung Ho; Sim, Taebo; Tae, Jin Sung; Lee, So Ha |
| 2020-07 | Sulfonamide-based 4-anilinoquinoline derivatives as novel dual Aurora kinase (AURKA/B) inhibitors: Synthesis, biological evaluation and in silico insights | Al-Sanea, Mohammad M.; Elkamhawy, Ahmed; Paik, Sora; Lee, Kyeong; El Kerdawy, Ahmed M.; Abbas, Bukhari Syed Nasir; Roh, Eun Joo; Eldehna, Wagdy M.; Elshemy, Heba A. H.; Bakr, Rania B.; Farahat, Ibrahim Ali; Alzarea, Abdulaziz, I; Alzarea, Sami, I; Alharbi, Khalid S.; Abdelgawad, Mohamed A. |
| 2013-03-15 | Synthesis and biological evaluation of 1-(2-hydroxy-3-phenyloxypropyl)piperazine derivatives as T-type calcium channel blockers | Park, Jung-eun; Ji, Wan Keun; Jang, Jae Wan; Pae, Ae Nim; Choi, Keehyun; Choi, Ki Hang; Kang, Jahyo; Roh, Eun Joo |
| 2015-11 | Synthesis and Biological Evaluation of 2-Phenylimino-5((5-phenylfuran-2-yl)methylene)thiazolidin-4-ones as IKK2 Inhibitors | Kim, Hee Sook; Shin, Min Jae; Lee, Byungho; Oh, Kwang-Seok; Choo, Hyunah; Pae, Ae Nim; Roh, Eun Joo; Nam, Ghilsoo |
| 2011-10-01 | Synthesis and biological evaluation of 4-piperidinecarboxylate and 4-piperidinecyanide derivatives for T-type calcium channel blockers | Woo, Hyun Min; Lee, Yun Suk; Roh, Eun Joo; Seo, Seon Hee; Song, Chi Man; Chung, Hye Jin; Pae, Ae Nim; Shin, Kye Jung |
| 2013-10-15 | Synthesis and biological evaluation of novel 3,4-diaryl lactam derivatives as triple reuptake inhibitors | Park, Jung-eun; Song, Chiman; Choi, Keehyun; Sim, Taebo; Moon, Bongjin; Roh, Eun Joo |
| 2019-01-01 | Synthesis and biological evaluation of novel 3-(quinolin-4-ylamino)benzenesulfonamidesAQ3 as carbonic anhydrase isoforms I and II inhibitors | Al-Sanea, Mohammad M.; Elkamhawy, Ahmed; Paik, Sora; Bua, Silvia; Lee, So Ha; Abdelgawad, Mohamed A.; Roh, Eun Joo; Eldehna, Wagdy M.; Supuran, Claudiu T. |
| 2018-01-20 | Synthesis and evaluation of 2-(3-arylureido)pyridines and 2-(3-arylureido)pyrazines as potential modulators of A beta-induced mitochondrial dysfunction in Alzheimer's disease | Elkamhawy, Ahmed; Park, Jung-eun; Hassan, Ahmed H. E.; Pae, Ae Nim; Lee, Jiyoun; Park, Beoung-Geon; Roh, Eun Joo |
| 2008-08-01 | Synthesis and evaluation of alpha,alpha'-disubstituted phenylacetate derivatives for T-type calcium channel blockers | Lee, Hyung Kook; Lee, Yun Suk; Roh, Eun Joo; Rhim, Hyewhon; Lee, Jae Yeol; Shin, Kye Jung |
| 2017-12-01 | Synthesis and evaluation of new pyridyl/pyrazinyl thiourea derivatives: Neuroprotection against amyloid-beta-induced toxicity | Park, Jung-eun; Elkamhawy, Ahmed; Hassan, Ahmed H. E.; Pae, Ae Nim; Lee, Jiyoun; Paik, Sora; Park, Beoung-Geon; Roh, Eun Joo |
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