Showing results 26 to 32 of 32
Issue Date | Title | Author(s) |
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2019-06 | Leveraging Compound Promiscuity to Identify Targetable Cysteines within the Kinome | Rao, Suman; Gurbani, Deepak; Du, Guangyan; Everley, Robert A.; Browne, Christopher M.; Chaikuad, Apirat; Tan, Li; Schroeder, Martin; Gondi, Sudershan; Ficarro, Scott B.; Sim, Taebo; Kim, Nam Doo; Berberich, Matthew J.; Knapp, Stefan; Marto, Jarrod A.; Westover, Kenneth D.; Sorger, Peter K.; Gray, Nathanael S. |
2022-02 | Novel Macrocyclic Peptidomimetics Targeting the Polo-Box Domain of Polo-Like Kinase 1 | Ryu, SeongShick; Park, Jung-Eun; Ham, Young Jin; Lim, Daniel C.; Kwiatkowski, Nicholas P.; Kim, Do-Hee; Bhunia, Debabrata; Kim, Nam Doo; Yaffe, Michael B.; Son, Woolim; Kim, Namkyoung; Choi, Tae-Ik; Swain, Puspanjali; Kim, Cheol-Hee; Lee, Jin-Young; Gray, Nathanael S.; Lee, Kyung S.; Sim, Tae Bo |
2012-02-18 | Rhodium-catalyzed reductive cyclization of 1,6-enynes and stereoselective synthesis of the putative structure of lucentamycin A and its stereoisomers | Ham, Young Jin; Yu, Hana; Kim, Nam Doo; Hah, Jung-Mi; Selim, Khalid B.; Choi, Hwan Geun; Sim, Taebo |
2018-09 | Structural and Atropisomeric Factors Governing the Selectivity of Pyrimido-benzodiazipinones as Inhibitors of Kinases and Bromodomains | Wang, Jinhua; Erazo, Tatiana; Ferguson, Fleur M.; Buckley, Dennis L.; Gomez, Nestor; Munoz-Guardiola, Pau; Dieguez-Martinez, Nora; Deng, Xianming; Hao, Mingfeng; Massefski, Walter; Fedorov, Oleg; Offei-Addo, Nana Kwaku; Park, Paul M.; Dai, Lingling; DiBona, Amy; Becht, Kelly; Kim, Nam Doo; McKeown, Michael R.; Roberts, Justin M.; Zhang, Jinwei; Sim, Taebo; Alessi, Dario R.; Bradner, James E.; Lizcano, Jose M.; Blacklow, Stephen C.; Qi, Jun; Xu, Xiang; Gray, Nathanael S. |
2019-08 | Synthesis and structure activity relationships of a series of 4-amino-1H-pyrazoles as covalent inhibitors of CDK14 | Ferguson, Fleur M.; Doctor, Zainab M.; Ficarro, Scott B.; Marto, Jarrod A.; Kim, Nam Doo; Sim, Taebo; Gray, Nathanael S. |
2014-07-30 | Targeting transcription regulation in cancer with a covalent CDK7 inhibitor | Kwiatkowski, Nicholas; Zhang, Tinghu; Rahl, Peter B.; Abraham, Brian J.; Reddy, Jessica; Ficarro, Scott B.; Dastur, Anahita; Amzallag, Arnaud; Ramaswamy, Sridhar; Tesar, Bethany; Jenkins, Catherine E.; Hannett, Nancy M.; McMillin, Douglas; Sanda, Takaomi; Sim, Taebo; Kim, Nam Doo; Look, Thomas; Mitsiades, Constantine S.; Weng, Andrew P.; Brown, Jennifer R.; Benes, Cyril H.; Marto, Jarrod A.; Young, Richard A.; Gray, Nathanael S. |
2014-01-03 | Therapeutic Targeting of Oncogenic K-Ras by a Covalent Catalytic Site Inhibitor | Lim, Sang Min; Westover, Kenneth D.; Ficarro, Scott B.; Harrison, Rane A.; Choi, Hwan Geun; Pacold, Michael E.; Carrasco, Martin; Hunter, John; Kim, Nam Doo; Xie, Ting; Sim, Taebo; Jaenne, Pasi A.; Meyerson, Matthew; Marto, Jarrod A.; Engen, John R.; Gray, Nathanael S. |