Showing results 1 to 30 of 33
Issue Date | Title | Author(s) |
---|---|---|
2014-11-24 | A new series of diarylamides possessing quinoline nucleus: Synthesis, in vitro anticancer activities, and kinase inhibitory effect | El-Gamal, Mohammed I.; Khan, Mohammad Ashrafuddin; Abdel-Maksoud, Mohammed S.; El-Din, Mahmoud M. Gamal; Oh, Chang-Hyun |
2022-09 | Antiamoebic Activity of Imidazothiazole Derivatives against Opportunistic Pathogen Acanthamoeba castellanii | Akbar, Noor; El-Gamal, Mohammed, I; Saeed, Balsam Qubais; Oh, Chang-Hyun; Abdel-Maksoud, Mohammed S.; Khan, Naveed Ahmed; Alharbi, Ahmad M.; Alfahemi, Hasan; Siddiqui, Ruqaiyyah |
2021-12 | Anticancer profile and anti-inflammatory effect of new N-(2-((4-(1,3-diphenyl-1H-pyrazol-4-yl)pyridine sulfonamide derivatives | Abdel-Maksoud, Mohammed S.; Hassan, Rasha Mohamed; El-Azzouny, Aida Abdel-Sattar; Aboul-Enein, Mohamed Nabil; Oh, Chang-Hyun |
2016-05 | Broad-spectrum antiproliferative activity of a series of 6-(4-fluorophenyl)-5-(2-substituted pyrimidin-4-yl)imidazo[2,1-b]thiazole derivatives | Abdel-Maksoud, Mohammed S.; El-Gamal, Mohammed I.; El-Din, Mahmoud M. Gamal; Kwak, Seong-Shin; Kim, Hyun-Il; Oh, Chang-Hyun |
2014-09 | Cell-Based Biological Evaluation of a New Bisamide FMS Kinase Inhibitor Possessing Pyrrolo[3,2-c]pyridine Scaffold | El-Gamal, Mohammed I.; Abdel-Maksoud, Mohammed S.; El-Din, Mahmoud M. Gamal; Yoo, Kyung Ho; Baek, Daejin; Oh, Chang-Hyun |
2023-01 | Design and synthesis of new adamantyl derivatives as promising antiproliferative agents | Shahin, Afnan, I; Zaraei, Seyed-Omar; AlKubaisi, Bilal O.; Ullah, Saif; Anbar, Hanan S.; El-Gamal, Randa; Menon, Varsha; Abdel-Maksoud, Mohammed S.; Oh, Chang-Hyun; El-Awady, Raafat; Gelsleichter, Nicolly Espindola; Pelletier, Julie; Sevigny, Jean; Iqbal, Jamshed; Al-Tel, Taleb H.; El-Gamal, Mohammed, I |
2017-02-15 | Design and synthesis of new RAF kinase-inhibiting antiproliferative quinoline derivatives. Part 2: Diarylurea derivatives | El-Gamal, Mohammed I.; Khan, Mohammad Ashrafuddin; Tarazi, Hamadeh; Abdel-Maksoud, Mohammed S.; El-Din, Mahmoud M. Gamal; Yoo, Kyung Ho; Oh, Chang-Hyun |
2020-06-01 | Design and synthesis of novel pyrrolo[2,3-b]pyridine derivatives targeting (V600E)BRAF | Abdel-Maksoud, Mohammed S.; Ali, Eslam M. H.; Ammar, Usama M.; Mersal, Karim I.; Yoo, Kyung Ho; Oh, Chang-Hyun |
2021-02-01 | Design, synthesis and anti-inflammatory activity of imidazol-5-yl pyridine derivatives as p38 alpha/MAPK14 inhibitor | Ali, Eslam M. H.; Abdel-Maksoud, Mohammed S.; Hassan, Rasha Mohamed; Mersal, Karim I.; Ammar, Usama M.; Se-In, Choi; He-Soo, Han; Kim, Hee-Kwon; Lee, Anna; Lee, Kyung-Tae; Oh, Chang-Hyun |
2019-12 | Design, synthesis, and anticancer activity of imidazo[2,1-b]oxazole-based RAF kinase inhibitors | Abdel-Maksoud, Mohammed S.; Ammar, Usama M.; El-Gamal, Mohammed I.; El-Din, Mahmoud M. Gamal; Mersal, Karim I.; Ali, Eslam M. H.; Yoo, Kyung Ho; Lee, Kyung-Tae; Oh, Chang-Hyun |
2012-07-01 | Design, synthesis, and antiproliferative activity of new 1H-pyrrolo[3,2-c]pyridine derivatives against melanoma cell lines. Part 2 | Jung, Myung-Ho; El-Gamal, Mohammed I.; Abdel-Maksoud, Mohammed S.; Sim, Taebo; Yoo, Kyung Ho; Oh, Chang-Hyun |
2021-01 | Design, synthesis, and biological evaluation of novel imidazole derivatives possessing terminal sulphonamides as potential BRAF(V600E) inhibitors | Ali, Eslam M. H.; Abdel-Maksoud, Mohammed S.; Ammar, Usama M.; Mersal, Karim, I; Yoo, Kyung Ho; Jooryeong, Park; Oh, Chang-Hyun |
2016-12 | Design, synthesis, and in vitro antiproliferative and kinase inhibitory effects of pyrimidinylpyrazole derivatives terminating with arylsulfonamido or cyclic sulfamide substituents | El-Din, Mahmoud M. Gamal; El-Gamal, Mohammed I.; Abdel-Maksoud, Mohammed S.; Yoo, Kyung Ho; Baek, Daejin; Choi, Jungseung; Lee, Huiseong; Oh, Chang-Hyun |
2021-04-05 | Design, synthesis, biological evaluation, and docking studies of novel (imidazol-5-yl)pyrimidine-based derivatives as dual BRAF(V600E)/p38 alpha inhibitors | Ali, Eslam M. H.; El-Telbany, Rania Farag A.; Abdel-Maksoud, Mohammed S.; Ammar, Usama M.; Mersal, Karim, I; Zaraei, Seyed-Omar; El-Gamal, Mohammed, I; Choi, Se-In; Lee, Kyung-Tae; Kim, Hee-Kwon; Lee, Kwan Hyi; Oh, Chang-Hyun |
2016-08-25 | Design, synthesis, broad-spectrum antiproliferative activity, and kinase inhibitory effect of triarylpyrazole derivatives possessing arylamides or arylureas moieties | El-Din, Mahmoud M. Gamal; El-Gamal, Mohammed I.; Abdel-Maksoud, Mohammed S.; Yoo, Kyung Ho; Oh, Chang-Hyun |
2019-01-01 | Design, synthesis, in vitro anticancer evaluation, kinase inhibitory effects, and pharmacokinetic profile of new 1,3,4-triarylpyrazole derivatives possessing terminal sulfonamide moiety | Abdel-Maksoud, Mohammed S.; El-Gamal, Mohammed I.; El-Din, Mahmoud M. Gamal; Oh, Chang Hyun |
2015-05-05 | Design, synthesis, in vitro antiproliferative evaluation, and kinase inhibitory effects of a new series of imidazo[2,1-b]thiazole derivatives | Abdel-Maksoud, Mohammed S.; Kim, Mi-Ryeong; El-Gamal, Mohammed I.; El-Din, Mahmoud M. Gamal; Tae, Jinsung; Choi, Hong Seok; Lee, Kyung-Tae; Yoo, Kyung Ho; Oh, Chang-Hyun |
2021-10 | Design, synthesis, in vitro determination and molecular docking studies of 4-(1-(tert-butyl)-3-phenyl-1H-pyrazol-4-yl) pyridine derivatives with terminal sulfonamide derivatives in LPS-induced RAW264.7 macrophage cells | Mersal, Karim I.; Abdel-Maksoud, Mohammed S.; Ali, Eslam M. H.; Ammar, Usama M.; Zaraei, Seyed-Omar; Kim, Jae-Min; Kim, Su-Yeon; Lee, Kyung-Tae; Lee, Kwan Hyi; Kim, Si-Won; Park, Hyun-Mee; Ji, Mi-Jung; Oh, Chang-Hyun |
2019-01-01 | Design, synthesis, in vitro potent antiproliferative activity, and kinase inhibitory effects of new triarylpyrazole derivatives possessing different heterocycle terminal moieties | El-Din, Mahmoud M. Gamal; El-Gamal, Mohammed I.; Abdel-Maksoud, Mohammed S.; Yoo, Kyung Ho; Oh, Chang-Hyun |
2021-11-15 | Discovery of first-in-class imidazothiazole-based potent and selective ErbB4 (HER4) kinase inhibitors | Zaraei, Seyed-Omar; Sbenati, Rawan M.; Alach, Nour N.; Anbar, Hanan S.; El-Gamal, Randa; Tarazi, Hamadeh; Shehata, Mahmoud K.; Abdel-Maksoud, Mohammed S.; Oh, Chang-Hyun; El-Gamal, Mohammed, I |
2021-05 | Discovery of New Imidazo[2,1-b]thiazole Derivatives as Potent Pan-RAF Inhibitors with Promising In Vitro and In Vivo Anti-melanoma Activity | Abdel-Maksoud, Mohammed S.; El-Gamal, Mohammed, I; Lee, Bong S.; El-Din, Mahmoud M. Gamal; Jeon, Hong R.; Kwon, Dow; Ammar, Usama M.; Mersal, Karim, I; Ali, Eslam M. H.; Lee, Kyung-Tae; Yoo, Kyung Ho; Han, Dong Keun; Lee, Jae Kyun; Kim, Garam; Choi, Hong Seok; Kwon, Young Jik; Lee, Kwan Hyi; Oh, Chang Hyun |
2023-12 | Evaluation of novel pyrazol-4-yl pyridine derivatives possessing arylsulfonamide tethers as c-Jun N-terminal kinase (JNK) inhibitors in leukemia cells | Mersal, Karim I.; Abdel-Maksoud, Mohammed S.; Ali, Eslam M. H.; Ammar, Usama M.; Zaraei, Seyed-Omar; Haque, Md Mamunul; Das, Tanuza; Hassan, Noha F.; Kim, Eunice EunKyeong; Lee, Jun-Seok; Park, Hajeung; Lee, Kwan Hyi; El-Gamal, Mohammed I.; Kim, Hee-Kwon; Ibrahim, Tamer M.; Oh, Chang-Hyun |
2019-03 | Mechanistic/mammalian target of rapamycin: Recent pathological aspects and inhibitors | Abdel-Maksoud, Mohammed S.; El-Gamal, Mohammed I.; Benhalilou, Dalia Reyane; Ashraf, Sandy; Mohammed, Shatha Abdulghaffar; Oh, Chang-Hyun |
2020-10-15 | Modification of imidazothiazole derivatives gives promising activity in B-Raf kinase enzyme inhibition; synthesis, in vitro studies and molecular docking | Ammar, Usama M.; Abdel-Maksoud, Mohammed S.; Mersal, Karim, I; Ali, Eslam M. H.; Yoo, Kyung Ho; Choi, Hong Seok; Lee, Jae Kyun; Cha, Sun Young; Oh, Chang-Hyun |
2013-08 | Recent Advances in the Research and Development of Marine Antimicrobial Peptides | El-Gamal, Mohammed I.; Abdel-Maksoud, Mohammed S.; Oh, Chang-Hyun |
2018-10-05 | Recent advances of RAF (rapidly accelerated fibrosarcoma) inhibitors as anti-cancer agents | Ammar, Usama M.; Abdel-Maksoud, Mohammed S.; Oh, Chang-Hyun |
2022-04 | Structural optimization of 4-(imidazol-5-yl)pyridine derivatives affords broad-spectrum anticancer agents with selective B-RAFV600E/p38α kinase inhibitory activity: Synthesis, in vitro assays and in silico study | Ibrahim Eslam Mohamed Hosny Ali; Karim Ibrahim Abdo Mersal; Ammar, Usama M.; Seyed Omar Zareei; Abdel-Maksoud, Mohammed S.; El-Gamal, Mohammed, I; Haque, Md Mamunul; Das, Tanuza; Kim, Eunice EunKyeong; Lee, Jun-Seok; LEE, KWAN HYI; Kim, Hee-Kwon; Oh, Chang Hyun |
2020-07 | Structural optimization of imidazothiazole derivatives affords a new promising series as B-Raf V600E inhibitors; synthesis, in vitro assay and in silico screening | Ammar, Usama M.; Abdel-Maksoud, Mohammed S.; Ali, Eslam M. H.; Mersal, Karim, I; Yoo, Kyung Ho; Oh, Chang-Hyun |
2015-04-15 | Synthesis and broad-spectrum antiproliferative activity of diarylamides and diarylureas possessing 1,3,4-oxadiazole derivatives | El-Din, Mahmoud M. Gamal; El-Gamal, Mohammed I.; Abdel-Maksoud, Mohammed S.; Yoo, Kyung Ho; Oh, Chang-Hyun |
2015-01-27 | Synthesis and in vitro antiproliferative activity of new 1,3,4-oxadiazole derivatives possessing sulfonamide moiety | El-Din, Mahmoud M. Gamal; El-Gamal, Mohammed I.; Abdel-Maksoud, Mohammed S.; Yoo, Kyung Ho; Oh, Chang-Hyun |