Showing results 1 to 6 of 6
Issue Date | Title | Author(s) |
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2017-09-15 | Characterization of a highly selective inhibitor of the Aurora kinases | Ferguson, Fleur M.; Doctor, Zainab M.; Chaikuad, Apirat; Sim, Taebo; Kim, Nam Doo; Knapp, Stefan; Gray, Nathanael S. |
2020-06 | Discovery of a selective inhibitor of doublecortin like kinase 1 | Ferguson, Fleur M.; Nabet, Behnam; Raghavan, Srivatsan; Liu, Yan; Leggett, Alan L.; Kuljanin, Miljan; Kalekar, Radha L.; Yang, Annan; He, Shuning; Wang, Jinhua; Ng, Raymond W. S.; Sulahian, Rita; Li, Lianbo; Poulin, Emily J.; Huang, Ling; Koren, Jost; Dieguez-Martinez, Nora; Espinosa, Sergio; Zeng, Zhiyang; Corona, Cesear R.; Vastall, James D.; Ohi, Ryoma; Sim, Tae Bo; Kim, Nam Doo; Harshbarger, Wayne; Lizcano, Jose M.; Robers, Matthew B.; Muthaswamy, Senthil; Lin, Charles Y.; Look, A. Thomas; Haigis, Kevin M.; Mancias, Joseph D.; Wolpin, Brian M.; Aguirre, Andrew J.; Hahn, William C.; Westover, Kenneth D.; Gray, Nathanael S. |
2016-10 | Discovery of a Series of 5,11-Dihydro-6H-benzo[e]pyrimido[5,4-b][1,4]diazepin-6-ones as Selective PI3K-delta/gamma Inhibitors | Ferguson, Fleur M.; Ni, Jing; Zhang, Tinghu; Tesar, Bethany; Sim, Taebo; Kim, Nam Doo; Deng, Xianming; Brown, Jennifer R.; Zhao, Jean J.; Gray, Nathanael S. |
2019-06 | Discovery of Covalent CDK14 Inhibitors with Pan-TAIRE Family Specificity | Ferguson, Fleur M.; Doctor, Zainab M.; Ficarro, Scott B.; Browne, Christopher M.; Marto, Jarrod A.; Johnson, Jared L.; Yaron, Tomer M.; Cantley, Lewis C.; Kim, Nam Doo; Sim, Taebo; Berberich, Matthew J.; Kalocsay, Marian; Sorger, Peter K.; Gray, Nathanael S. |
2018-09 | Structural and Atropisomeric Factors Governing the Selectivity of Pyrimido-benzodiazipinones as Inhibitors of Kinases and Bromodomains | Wang, Jinhua; Erazo, Tatiana; Ferguson, Fleur M.; Buckley, Dennis L.; Gomez, Nestor; Munoz-Guardiola, Pau; Dieguez-Martinez, Nora; Deng, Xianming; Hao, Mingfeng; Massefski, Walter; Fedorov, Oleg; Offei-Addo, Nana Kwaku; Park, Paul M.; Dai, Lingling; DiBona, Amy; Becht, Kelly; Kim, Nam Doo; McKeown, Michael R.; Roberts, Justin M.; Zhang, Jinwei; Sim, Taebo; Alessi, Dario R.; Bradner, James E.; Lizcano, Jose M.; Blacklow, Stephen C.; Qi, Jun; Xu, Xiang; Gray, Nathanael S. |
2019-08 | Synthesis and structure activity relationships of a series of 4-amino-1H-pyrazoles as covalent inhibitors of CDK14 | Ferguson, Fleur M.; Doctor, Zainab M.; Ficarro, Scott B.; Marto, Jarrod A.; Kim, Nam Doo; Sim, Taebo; Gray, Nathanael S. |