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Showing results 1 to 28 of 28

Issue DateTitleAuthor(s)
2010-08-12A Type-II Kinase Inhibitor Capable of Inhibiting the T315I "Gatekeeper" Mutant of Bcr-AblChoi, Hwan Geun; Ren, Pingda; Adrian, Francisco; Sun, Fangxian; Lee, Hyun Soo; Wang, Xia; Ding, Qiang; Zhang, Guobao; Xie, Yongping; Zhang, Jianming; Liu, Yi; Tuntland, Tove; Warmuth, Markus; Manley, Paul W.; Mestan, Juergen; Gray, Nathanael S.; Sim, Taebo
2017-09-15Characterization of a highly selective inhibitor of the Aurora kinasesFerguson, Fleur M.; Doctor, Zainab M.; Chaikuad, Apirat; Sim, Taebo; Kim, Nam Doo; Knapp, Stefan; Gray, Nathanael S.
2017-01Covalent Guanosine Mimetic Inhibitors of G12C KRASXiong, Yuan; Lu, Jia; Hunter, John; Li, Lianbo; Scott, David; Choi, Hwan Geun; Lim, Sang Min; Manandhar, Anuj; Gondi, Sudershan; Sim, Taebo; Westover, Kenneth D.; Gray, Nathanael S.
2012-08-15Development of 'DFG-out' inhibitors of gatekeeper mutant kinasesChoi, Hwan Geun; Zhang, Jianming; Weisberg, Ellen; Griffin, James D.; Sim, Taebo; Gray, Nathanael S.
2019-06Development of a Selective CDK7 Covalent Inhibitor Reveals Predominant Cell-Cycle PhenotypeOlson, Calla M.; Liang, Yanke; Leggett, Alan; Park, Woojun D.; Li, Lianbo; Mills, Caitlin E.; Elsarrag, Selma Z.; Ficarro, Scott B.; Zhang, Tinghu; Duester, Robert; Geyer, Matthias; Sim, Taebo; Marto, Jarrod A.; Sorger, Peter K.; Westover, Ken D.; Lin, Charles Y.; Kwiatkowski, Nicholas; Gray, Nathanael S.
2016-08Development of Chemical Probes for Investigation of Salt-Inducible Kinase Function in VivoSundberg, Thomas B.; Liang, Yanke; Wu, Huixian; Choi, Hwan Geun; Kim, Nam Doo; Sim, Taebo; Johannessen, Liv; Petrone, Adam; Khor, Bernard; Graham, Daniel B.; Latorre, Isabel J.; Phillips, Andrew J.; Schreiber, Stuart L.; Perez, Jose; Shamji, Alykhan F.; Gray, Nathanael S.; Xavier, Ramnik J.
2014-11-11Development of covalent inhibitors that can overcome resistance to first-generation FGFR kinase inhibitorsTan, Li; Wang, Jun; Tanizaki, Junko; Huang, Zhifeng; Aref, Amir R.; Rusan, Maria; Zhu, Su-Jie; Zhang, Yiyun; Ercan, Dalia; Liao, Rachel G.; Capelletti, Marzia; Zhou, Wenjun; Hur, Wooyoung; Kim, NamDoo; Sim, Taebo; Gaudet, Suzanne; Barbie, David A.; Yeh, Jing-Ruey Joanna; Yun, Cai-Hong; Hammerman, Peter S.; Mohammadi, Moosa; Jaenne, Pasi A.; Gray, Nathanael S.
2018-06Development of Highly Potent and Selective Steroidal Inhibitors and Degraders of CDK8Hatcher, John M.; Wang, Eric S.; Johannessen, Liv; Kwiatkowski, Nicholas; Sim, Taebo; Gray, Nathanael S.
2016-05Discovery of a Highly Potent and Selective Indenoindolone Type 1 Pan-FLT3 InhibitorHatcher, John M.; Weisberg, Ellen; Sim, Taebo; Stone, Richard M.; Liu, Suiyang; Griffin, James D.; Gray, Nathanael S.
2020-06Discovery of a selective inhibitor of doublecortin like kinase 1Ferguson, Fleur M.; Nabet, Behnam; Raghavan, Srivatsan; Liu, Yan; Leggett, Alan L.; Kuljanin, Miljan; Kalekar, Radha L.; Yang, Annan; He, Shuning; Wang, Jinhua; Ng, Raymond W. S.; Sulahian, Rita; Li, Lianbo; Poulin, Emily J.; Huang, Ling; Koren, Jost; Dieguez-Martinez, Nora; Espinosa, Sergio; Zeng, Zhiyang; Corona, Cesear R.; Vastall, James D.; Ohi, Ryoma; Sim, Tae Bo; Kim, Nam Doo; Harshbarger, Wayne; Lizcano, Jose M.; Robers, Matthew B.; Muthaswamy, Senthil; Lin, Charles Y.; Look, A. Thomas; Haigis, Kevin M.; Mancias, Joseph D.; Wolpin, Brian M.; Aguirre, Andrew J.; Hahn, William C.; Westover, Kenneth D.; Gray, Nathanael S.
2016-10Discovery of a Series of 5,11-Dihydro-6H-benzo[e]pyrimido[5,4-b][1,4]diazepin-6-ones as Selective PI3K-delta/gamma InhibitorsFerguson, Fleur M.; Ni, Jing; Zhang, Tinghu; Tesar, Bethany; Sim, Taebo; Kim, Nam Doo; Deng, Xianming; Brown, Jennifer R.; Zhao, Jean J.; Gray, Nathanael S.
2019-06Discovery of Covalent CDK14 Inhibitors with Pan-TAIRE Family SpecificityFerguson, Fleur M.; Doctor, Zainab M.; Ficarro, Scott B.; Browne, Christopher M.; Marto, Jarrod A.; Johnson, Jared L.; Yaron, Tomer M.; Cantley, Lewis C.; Kim, Nam Doo; Sim, Taebo; Berberich, Matthew J.; Kalocsay, Marian; Sorger, Peter K.; Gray, Nathanael S.
2015-12-10Discovery of Inhibitors That Overcome the G1202R Anaplastic Lymphoma Kinase Resistance MutationHatcher, John M.; Bahcall, Magda; Choi, Hwan Geun; Gao, Yang; Sim, Taebo; George, Rani; Jaenne, Pasi A.; Gray, Nathanael S.
2012-01-27Discovery of Potent and Selective Covalent Inhibitors of JNKZhang, Tinghu; Inesta-Vaquera, Francisco; Niepel, Mario; Zhang, Jianming; Ficarro, Scott B.; Machleidt, Thomas; Xie, Ting; Marto, Jarrod A.; Kim, NamDoo; Sim, Taebo; Laughlin, John D.; Park, Hajeung; LoGrasso, Philip V.; Patricelli, Matt; Nomanbhoy, Tyzoon K.; Sorger, Peter K.; Alessi, Dario R.; Gray, Nathanael S.
2015-01-08Discovery of Type II Inhibitors of TGF beta-Activated Kinase 1 (TAK1) and Mitogen-Activated Protein Kinase Kinase Kinase Kinase 2 (MAP4K2)Tan, Li; Nomanbhoy, Tyzoon; Gurbani, Deepak; Patricelli, Matthew; Hunter, John; Geng, Jiefei; Herhaus, Lina; Zhang, Jianming; Pauls, Eduardo; Ham, Youngjin; Choi, Hwan Geun; Xie, Ting; Deng, Xianming; Buhrlage, Sara J.; Sim, Taebo; Cohen, Philip; Sapkota, Gopal; Westover, Kenneth D.; Gray, Nathanael S.
2010-10-14Expanding the Diversity of Allosteric Ber-Abl InhibitorsDeng, Xianming; Okram, Barun; Ding, Qiang; Zhang, Jianming; Choi, Yongmun; Adrian, Francisco J.; Wojciechowski, Amy; Zhang, Guobao; Che, Jianwei; Bursulaya, Badry; Cowan-Jacob, Sandra W.; Rummel, Gabriele; Sim, Taebo; Gray, Nathanael S.
2018-09-27First SAR Study for Overriding NRAS Mutant Driven Acute Myeloid LeukemiaCho, Hanna; Shin, Injae; Ju, Eunhye; Choi, Seunghye; Hur, Wooyoung; Kim, Haelee; Hong, Eunmi; Kim, Nam Doo; Choi, Hwan Geun; Gray, Nathanael S.; Sim, Taebo
2017-01-01Identification of Existing Drugs That Effectively Target NTRK1 and ROS1 Rearrangements in Lung CancerChong, Curtis R.; Bahcall, Magda; Capelletti, Marzia; Kosaka, Takayuki; Ercan, Dalia; Sim, Taebo; Sholl, Lynette M.; Nishino, Mizuki; Johnson, Bruce E.; Gray, Nathanael S.; Janne, Pasi A.
2015-05-14Identification of novel therapeutic targets in acute leukemias with NRAS mutations using a pharmacologic approachNonami, Atsushi; Sattler, Martin; Weisberg, Ellen; Liu, Qingsong; Zhang, Jianming; Patricelli, Matthew P.; Christie, Amanda L.; Saur, Amy M.; Kohl, Nancy E.; Kung, Andrew L.; Yoon, Hojong; Sim, Taebo; Gray, Nathanael S.; Griffin, James D.
2019-06Leveraging Compound Promiscuity to Identify Targetable Cysteines within the KinomeRao, Suman; Gurbani, Deepak; Du, Guangyan; Everley, Robert A.; Browne, Christopher M.; Chaikuad, Apirat; Tan, Li; Schroeder, Martin; Gondi, Sudershan; Ficarro, Scott B.; Sim, Taebo; Kim, Nam Doo; Berberich, Matthew J.; Knapp, Stefan; Marto, Jarrod A.; Westover, Kenneth D.; Sorger, Peter K.; Gray, Nathanael S.
2022-02Novel Macrocyclic Peptidomimetics Targeting the Polo-Box Domain of Polo-Like Kinase 1Ryu, SeongShick; Park, Jung-Eun; Ham, Young Jin; Lim, Daniel C.; Kwiatkowski, Nicholas P.; Kim, Do-Hee; Bhunia, Debabrata; Kim, Nam Doo; Yaffe, Michael B.; Son, Woolim; Kim, Namkyoung; Choi, Tae-Ik; Swain, Puspanjali; Kim, Cheol-Hee; Lee, Jin-Young; Gray, Nathanael S.; Lee, Kyung S.; Sim, Tae Bo
2014-12Pharmacological targeting of the pseudokinase Her3Xie, Ting; Lim, Sang Min; Westover, Kenneth D.; Dodge, Michael E.; Ercan, Dalia; Ficarro, Scott B.; Udayakumar, Durga; Gurbani, Deepak; Tae, Hyun Seop; Riddle, Steven M.; Sim, Taebo; Marto, Jarrod A.; Jaenne, Pasi A.; Crews, Craig M.; Gray, Nathanael S.
2018-09Structural and Atropisomeric Factors Governing the Selectivity of Pyrimido-benzodiazipinones as Inhibitors of Kinases and BromodomainsWang, Jinhua; Erazo, Tatiana; Ferguson, Fleur M.; Buckley, Dennis L.; Gomez, Nestor; Munoz-Guardiola, Pau; Dieguez-Martinez, Nora; Deng, Xianming; Hao, Mingfeng; Massefski, Walter; Fedorov, Oleg; Offei-Addo, Nana Kwaku; Park, Paul M.; Dai, Lingling; DiBona, Amy; Becht, Kelly; Kim, Nam Doo; McKeown, Michael R.; Roberts, Justin M.; Zhang, Jinwei; Sim, Taebo; Alessi, Dario R.; Bradner, James E.; Lizcano, Jose M.; Blacklow, Stephen C.; Qi, Jun; Xu, Xiang; Gray, Nathanael S.
2013-12Structural determinants for ERK5 (MAPK7) and leucine rich repeat kinase 2 activities of benzo[e]pyrimido-[5,4-b]diazepine-6(11H)-onesDeng, Xianming; Elkins, Jonathan M.; Zhang, Jinwei; Yang, Qingkai; Erazo, Tatiana; Gomez, Nestor; Choi, Hwan Geun; Wang, Jinhua; Dzamko, Nicolas; Lee, Jiing-Dwan; Sim, Taebo; Kim, NamDoo; Alessi, Dario R.; Lizcano, Jose M.; Knapp, Stefan; Gray, Nathanael S.
2019-08Synthesis and structure activity relationships of a series of 4-amino-1H-pyrazoles as covalent inhibitors of CDK14Ferguson, Fleur M.; Doctor, Zainab M.; Ficarro, Scott B.; Marto, Jarrod A.; Kim, Nam Doo; Sim, Taebo; Gray, Nathanael S.
2010-01-28Targeting Bcr-Abl by combining allosteric with ATP-binding-site inhibitorsZhang, Jianming; Adrian, Francisco J.; Jahnke, Wolfgang; Cowan-Jacob, Sandra W.; Li, Allen G.; Iacob, Roxana E.; Sim, Taebo; Powers, John; Dierks, Christine; Sun, Fangxian; Guo, Gui-Rong; Ding, Qiang; Okram, Barun; Choi, Yongmun; Wojciechowski, Amy; Deng, Xianming; Liu, Guoxun; Fendrich, Gabriele; Strauss, Andre; Vajpai, Navratna; Grzesiek, Stephan; Tuntland, Tove; Liu, Yi; Bursulaya, Badry; Azam, Mohammad; Manley, Paul W.; Engen, John R.; Daley, George Q.; Warmuth, Markus; Gray, Nathanael S.
2014-07-30Targeting transcription regulation in cancer with a covalent CDK7 inhibitorKwiatkowski, Nicholas; Zhang, Tinghu; Rahl, Peter B.; Abraham, Brian J.; Reddy, Jessica; Ficarro, Scott B.; Dastur, Anahita; Amzallag, Arnaud; Ramaswamy, Sridhar; Tesar, Bethany; Jenkins, Catherine E.; Hannett, Nancy M.; McMillin, Douglas; Sanda, Takaomi; Sim, Taebo; Kim, Nam Doo; Look, Thomas; Mitsiades, Constantine S.; Weng, Andrew P.; Brown, Jennifer R.; Benes, Cyril H.; Marto, Jarrod A.; Young, Richard A.; Gray, Nathanael S.
2014-01-03Therapeutic Targeting of Oncogenic K-Ras by a Covalent Catalytic Site InhibitorLim, Sang Min; Westover, Kenneth D.; Ficarro, Scott B.; Harrison, Rane A.; Choi, Hwan Geun; Pacold, Michael E.; Carrasco, Martin; Hunter, John; Kim, Nam Doo; Xie, Ting; Sim, Taebo; Jaenne, Pasi A.; Meyerson, Matthew; Marto, Jarrod A.; Engen, John R.; Gray, Nathanael S.
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