Browsing byAuthorRoh, Eun Joo
Showing results 1 to 30 of 66
| Issue Date | Title | Author(s) |
|---|---|---|
| 2022-06 | 2-(3-Bromophenyl)-8-fluoroquinazoline-4-carboxylic Acid as a Novel and Selective Aurora A Kinase Inhibitory Lead with Apoptosis Properties: Design, Synthesis, In Vitro and In Silico Biological Evaluation | Elsherbeny, Mohamed H.; Ammar, Usama M.; Abdellattif, Magda H.; Abourehab, Mohammed A. S.; Abdeen, Ahmed; Ibrahim, Samah F.; Abdelrahaman, Doaa; Mady, Wessam; Roh, Eun Joo; Elkamhawy, Ahmed |
| 2022-07 | AF8c, a Multi-Kinase Inhibitor Induces Apoptosis by Activating DR5/Nrf2 via ROS in Colorectal Cancer Cells | Jeong, Soyeon; Farag, Ahmed K.; Yun, Hye Kyeong; Jeong, Yoon A.; Kim, Dae Yeong; Jo, Min Jee; Park, Seong Hye; Kim, Bo Ram; Kim, Jung Lim; Kim, Bu Gyeom; Lee, Dae-Hee; Roh, Eun Joo; Oh, Sang Cheul |
| 2019-10 | AF8c, a pan-ErbB family inhibitor induces apoptotic cell death by stimulating DR5/Nrf2 via ROS in colorectal cancer cells | Jeong, Soyeon; Farag, Ahmed Karam; Yun, Hye Kyeong; Jeong, Yoon A.; Kim, Dae Yeong; Jo, Min Jee; Park, Seong Hye; Kim, Bo Ram; Kim, Jung Lim; Lee, Dae-Hee; Roh, Eun Joo; Oh, Sang Cheul |
| 2010-02-01 | Caffeine-Mediated Inhibition of Calcium Release Channel Inositol 1,4,5-Trisphosphate Receptor Subtype 3 Blocks Glioblastoma Invasion and Extends Survival | Kang, Sang Soo; Han, Kyung-Seok; Ku, Bo Mi; Lee, Yeon Kyung; Hong, Jinpyo; Shin, Hye Young; Almonte, Antoine G.; Woo, Dong Ho; Brat, Daniel J.; Hwang, Eun Mi; Yoo, Seung Hyun; Chung, Chun Kee; Park, Sung-Hye; Paek, Sun Ha; Roh, Eun Joo; Lee, Sung Joong; Park, Jae-Yong; Traynelis, Stephen F.; Lee, C. Justin |
| 2019-01 | Death-associated protein kinase (DAPK) family modulators: Current and future therapeutic outcomes | Farag, Ahmed Karam; Roh, Eun Joo |
| 2015-07 | Design and Synthesis of New [1,2,3]Triazolo[4,5-d]pyrimidine Derivatives as Potential Antiproliferative Agents | Elkamhawy, Ahmed; Al-Sanea, Mohammad M.; Song, Chiman; Sim, Taebo; Roh, Eun Joo |
| 2022-07 | Design, Synthesis and Biological Evaluation of 1,3,5-Triazine Derivatives Targeting hA(1) and hA(3) Adenosine Receptor | Park, Sujin; Ahn, Yujin; Kim, Yongchan; Roh, Eun Joo; Lee, Yoonji; Han, Chaebin; Yoo, Hee Min; Yu, Jinha |
| 2018-09-05 | Design, synthesis and biological evaluation of novel thiazolidinedione derivatives as irreversible allosteric IKK-beta modulators | Elkamhawy, Ahmed; Kim, Nam Youn; Hassan, Ahmed H. E.; Park, Jung-eun; Yang, Jeong-Eun; Oh, Kwang-Seok; Lee, Byung Ho; Lee, Mi Young; Shin, Kye Jung; Lee, Kyung-Tae; Hur, Wooyoung; Roh, Eun Joo |
| 2018-12-15 | Design, synthesis, and biological evaluation of novel aminopyrimidinylisoindolines as AXL kinase inhibitors | Choi, Min Jung; Roh, Eun Joo; Hur, Wooyoung; Lee, So Ha; Sim, Taebo; Oh, Chang-Hyun; Lee, Sun-Hwa; Kim, Jong Seung; Yoo, Kyung Ho |
| 2022-09 | Design, synthesis, and biological evaluation of pseudo-bicyclic pyrimidine-based compounds as potential EGFR inhibitors | Farag, Ahmed Karam; Ahn, Byung Sun; Yoo, Je Sik; Karam, Reham; Roh, Eun Joo |
| 2017-06-15 | Design, synthesis, biological evaluation and molecular modelling of 2-(2-aryloxyphenyl)-1,4-dihydroisoquinolin-3(2H)-ones: A novel class of TSPO ligands modulating amyloid-beta-induced mPTP opening | Elkamhawy, Ahmed; Park, Jung-eun; Hassan, Ahmed H. E.; Pae, Ae Nim; Lee, Jiyoun; Park, Beoung-Geon; Paik, Sora; Do, Jimin; Park, Jong-Hyun; Park, Ki Duk; Moon, Bongjin; Park, Woo Kyu; Cho, Heeyeong; Jeong, Dae Young; Roh, Eun Joo |
| 2014-05-03 | Determination of Edible Vegetable Oil Adulterants in Sesame Oil Using H-1 Nuclear Magnetic Resonance Spectroscopy | Nam, Yun Sik; Noh, Kown-Chul; Roh, Eun Joo; Keum, Gyochang; Lee, Yeonhee; Lee, Kang-Bong |
| 2021-01-14 | Development and Therapeutic Potential of NUAKs Inhibitors | Faisal, Muhammad; Kim, Jae Ho; Yoo, Kyung Ho; Roh, Eun Joo; Hong, Soon Sun; Lee, So Ha |
| 2021-09 | Development of New Meridianin/Leucettine-Derived Hybrid Small Molecules as Nanomolar Multi-Kinase Inhibitors with Antitumor Activity | Elsherbeny, Mohamed H.; Elkamhawy, Ahmed; Nada, Hossam; Abdellattif, Magda H.; Lee, Kyeong; Roh, Eun Joo |
| 2008-10 | Development of selective blockers for Ca2+-activated Cl- channel using Xenopus laevis oocytes with an improved drug screening strategy | Oh, Soo-Jin; Park, Jung Hwan; Han, Sungyu; Lee, Jae Kyun; Roh, Eun Joo; Lee, C. Justin |
| 2023-12 | Diabetes mellitus: Classification, mediators, and complications; A gate to identify potential targets for the development of new effective treatments | Antar, Samar A.; Ashour, Nada A.; Sharaky, Marwa; Khattab, Muhammad; Ashour, Naira A.; Zaid, Roaa T.; Roh, Eun Joo; Elkamhawy, Ahmed; Al-Karmalawy, Ahmed A. |
| 2020-10 | Diarylurea derivatives comprising 2,4-diarylpyrimidines: Discovery of novel potential anticancer agents via combined failed-ligands repurposing and molecular hybridization approaches | Farag, Ahmed Karam; Hassan, Ahmed H. E.; Chung, Kyung-Sook; Lee, Jeong-Hun; Gil, Hyo-Sun; Lee, Kyung-Tae; Roh, Eun Joo |
| 2017-03-10 | Discovery of 1-(3-(benzyloxy)pyridin-2-yl)-3-(2-(piperazin-1-yl)ethyl)urea: A new modulator for amyloid beta-induced mitochondrial dysfunction | Elkamhawy, Ahmed; Park, Jung-Eun; Hassan, Ahmed H. E.; Ra, Hyunhwa; Pae, Ae Nim; Lee, Jiyoun; Park, Beoung-Geon; Moon, Bongjin; Park, Hyun-Mee; Roh, Eun Joo |
| 2021-11 | Discovery of 3,4-dichloro-N-(1H-indol-5-yl)benzamide: A highly potent, selective, and competitive hMAO-B inhibitor with high BBB permeability and action | Elkamhawy, Ahmed; Kim, Hyeon Jeong; Elsherbeny, Mohamed H.; Paik, Sora; Park, Jong-Hyun; Gotina, Lizaveta; Abdellattif, Magda H.; Gouda, Noha A.; Cho, Jungsook; Lee, Kyeong; Pae, Ae Nim; Park, Ki Duk; Roh, Eun Joo |
| 2016-01-02 | Discovery of a broad spectrum antiproliferative agent with selectivity for DDR1 kinase: cell line-based assay, kinase panel, molecular docking, and toxicity studies | Elkamhawy, Ahmed; Park, Jung-eun; Cho, Nam-Chul; Sim, Taebo; Pae, Ae Nim; Roh, Eun Joo |
| 2020-01 | Discovery of N-(1-(3-fluorobenzoyl)-1H-indol-5-yl)pyrazine-2-carboxamide: a novel, selective, and competitive indole-based lead inhibitor for human monoamine oxidase B | Elkamhawy, Ahmed; Paik, Sora; Kim, Hyeon Jeong; Park, Jong-Hyun; Londhe, Ashwini M.; Lee, Kyeong; Pae, Ae Nim; Park, Ki Duk; Roh, Eun Joo |
| 2024-03 | Discovery of N-benzylbenzamide-based allosteric inhibitors of Aurora kinase A | Lee, Hyomin; Kim, Euijung; Hwang, Narae; Yoo, Jesik; Nam, Yunju; Hwang, Injeoung; Park, Jin-Gyeong; Park, Sang-Eun; Chung, Kyung-Sook; Chung, Hwan Won; Song, Chiman; Ji, Mi-Jung; Park, Hyun-Mee; Lee, In-Kyun; Lee, Kyung-Tae; Roh, Eun Joo; Hur, Wooyoung |
| 2011-05-15 | Discovery of piperidinyl aminopyrimidine derivatives as IKK-2 inhibitors | Kim, Sora; Jung, Jin Kyo; Lee, Hyo Seon; Kim, Youngjae; Kim, Jiyoon; Choi, Kihang; Baek, Du-Jong; Moon, Bongjin; Oh, Kwang-Seok; Lee, Byung Ho; Shin, Kye Jung; Pae, Ae Nim; Nam, Ghilsoo; Roh, Eun Joo; Cho, Yong Seo; Choo, Hyunah |
| 2015-10-20 | Discovery of potent and selective cytotoxic activity of new quinazoline-ureas against TMZ-resistant glioblastoma multiforme (GBM) | Elkamhawy, Ahmed; Viswanath, Ambily Nath Indu; Pae, Ae Nim; Kim, Hyeon Young; Heo, Jin-Chul; Park, Woo-Kyu; Lee, Chong-Ock; Yang, Heekyoung; Kim, Kang Ho; Nam, Do-Hyun; Seol, Ho Jun; Cho, Heeyeong; Roh, Eun Joo |
| 2012-09-01 | Discovery of potent and selective rhodanine type IKK beta inhibitors by hit-to-lead strategy | Song, Hyeseung; Lee, Yun Suk; Roh, Eun Joo; Seo, Jae Hong; Oh, Kwang-Seok; Lee, Byung Ho; Han, Hogyu; Shin, Kye Jung |
| 2019-05 | EGFR inhibitors from cancer to inflammation: Discovery of 4-fluoro-N-(4-(3-(trifluoromethyl)phenoxy)pyrimidin-5-yl)benzamide as a novel anti-inflammatory EGFR inhibitor | Elkamhawy, Ahmed; Hassan, Ahmed H. E.; Paik, Sora; Lee, Yong Sup; Lee, Hwi-Ho; Shin, Ji-Sun; Lee, Kyung-Tae; Roh, Eun Joo |
| 2019-01-15 | First-in-class DAPK1/CSF1R dual inhibitors: Discovery of 3,5-dimethoxy-N-(4-(4-methoxyphenoxy)-24(6-morpholinopyridin-3-yl)amino) pyrimidin-5-yl)benzamide as a potential anti-tauopathies agent | Farag, Ahmed Karam; Hassan, Ahmed H. E.; Jeong, Hyeanjeong; Kwon, Youngji; Choi, Jin Gyu; Oh, Myung Sook; Park, Ki Duk; Kim, Yun Kyung; Roh, Eun Joo |
| 2008-05 | Functional human 5-HT6 receptor assay for high throughput screening of chemical ligands and binding proteins | Kim, Hyun-Ji; Yun, Hyung-Mun; Kim, Taehyun; Nam, Ghilsoo; Roh, Eun Joo; Kostenis, Evi; Choo, Hea-Young Park; Pae, Ae Nim; Rhim, Hyewhon |
| 2017-11 | Hit discovery of 4-amino-N-(4-(3-(trifluoromethyl)phenoxy)pyrimidin-5-yl)benzamide: A novel EGFR inhibitor from a designed small library | Elkamhawy, Ahmed; Paik, Sora; Hassan, Ahmed H. E.; Lee, Yong Sup; Roh, Eun Joo |
| 2022-09 | Identification of Novel Aryl Carboxamide Derivatives as Death-Associated Protein Kinase 1 (DAPK1) Inhibitors with Anti-Proliferative Activities: Design, Synthesis, In Vitro, and In Silico Biological Studies | Elkamhawy, Ahmed; Paik, Sora; Ali, Eslam M. H.; Hassan, Ahmed H. E.; Kang, So Jin; Lee, Kyeong; Roh, Eun Joo |
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