Showing results 1 to 6 of 6
Issue Date | Title | Author(s) |
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2017-01 | Covalent Guanosine Mimetic Inhibitors of G12C KRAS | Xiong, Yuan; Lu, Jia; Hunter, John; Li, Lianbo; Scott, David; Choi, Hwan Geun; Lim, Sang Min; Manandhar, Anuj; Gondi, Sudershan; Sim, Taebo; Westover, Kenneth D.; Gray, Nathanael S. |
2020-06 | Discovery of a selective inhibitor of doublecortin like kinase 1 | Ferguson, Fleur M.; Nabet, Behnam; Raghavan, Srivatsan; Liu, Yan; Leggett, Alan L.; Kuljanin, Miljan; Kalekar, Radha L.; Yang, Annan; He, Shuning; Wang, Jinhua; Ng, Raymond W. S.; Sulahian, Rita; Li, Lianbo; Poulin, Emily J.; Huang, Ling; Koren, Jost; Dieguez-Martinez, Nora; Espinosa, Sergio; Zeng, Zhiyang; Corona, Cesear R.; Vastall, James D.; Ohi, Ryoma; Sim, Tae Bo; Kim, Nam Doo; Harshbarger, Wayne; Lizcano, Jose M.; Robers, Matthew B.; Muthaswamy, Senthil; Lin, Charles Y.; Look, A. Thomas; Haigis, Kevin M.; Mancias, Joseph D.; Wolpin, Brian M.; Aguirre, Andrew J.; Hahn, William C.; Westover, Kenneth D.; Gray, Nathanael S. |
2015-01-08 | Discovery of Type II Inhibitors of TGF beta-Activated Kinase 1 (TAK1) and Mitogen-Activated Protein Kinase Kinase Kinase Kinase 2 (MAP4K2) | Tan, Li; Nomanbhoy, Tyzoon; Gurbani, Deepak; Patricelli, Matthew; Hunter, John; Geng, Jiefei; Herhaus, Lina; Zhang, Jianming; Pauls, Eduardo; Ham, Youngjin; Choi, Hwan Geun; Xie, Ting; Deng, Xianming; Buhrlage, Sara J.; Sim, Taebo; Cohen, Philip; Sapkota, Gopal; Westover, Kenneth D.; Gray, Nathanael S. |
2019-06 | Leveraging Compound Promiscuity to Identify Targetable Cysteines within the Kinome | Rao, Suman; Gurbani, Deepak; Du, Guangyan; Everley, Robert A.; Browne, Christopher M.; Chaikuad, Apirat; Tan, Li; Schroeder, Martin; Gondi, Sudershan; Ficarro, Scott B.; Sim, Taebo; Kim, Nam Doo; Berberich, Matthew J.; Knapp, Stefan; Marto, Jarrod A.; Westover, Kenneth D.; Sorger, Peter K.; Gray, Nathanael S. |
2014-12 | Pharmacological targeting of the pseudokinase Her3 | Xie, Ting; Lim, Sang Min; Westover, Kenneth D.; Dodge, Michael E.; Ercan, Dalia; Ficarro, Scott B.; Udayakumar, Durga; Gurbani, Deepak; Tae, Hyun Seop; Riddle, Steven M.; Sim, Taebo; Marto, Jarrod A.; Jaenne, Pasi A.; Crews, Craig M.; Gray, Nathanael S. |
2014-01-03 | Therapeutic Targeting of Oncogenic K-Ras by a Covalent Catalytic Site Inhibitor | Lim, Sang Min; Westover, Kenneth D.; Ficarro, Scott B.; Harrison, Rane A.; Choi, Hwan Geun; Pacold, Michael E.; Carrasco, Martin; Hunter, John; Kim, Nam Doo; Xie, Ting; Sim, Taebo; Jaenne, Pasi A.; Meyerson, Matthew; Marto, Jarrod A.; Engen, John R.; Gray, Nathanael S. |