2019-06 | Development of a Selective CDK7 Covalent Inhibitor Reveals Predominant Cell-Cycle Phenotype | Olson, Calla M.; Liang, Yanke; Leggett, Alan; Park, Woojun D.; Li, Lianbo; Mills, Caitlin E.; Elsarrag, Selma Z.; Ficarro, Scott B.; Zhang, Tinghu; Duester, Robert; Geyer, Matthias; Sim, Taebo; Marto, Jarrod A.; Sorger, Peter K.; Westover, Ken D.; Lin, Charles Y.; Kwiatkowski, Nicholas; Gray, Nathanael S. |
2019-01-01 | Identification of 1H-pyrazolo[3,4-b]pyridine derivatives as potent ALK-L1196M inhibitors | Nam, Yunju; Hwang, Dongkeun; Kim, Namdoo; Seo, Hong-Seog; Selim, Khalid B.; Sim, Taebo |
2019-05 | A Bcr-Abl Inhibitor GNF-2 Attenuates Inflammatory Activation of Glia and Chronic Pain | Song, Gyun Jee; Rahman, Md Habibur; Jha, Mithilesh Kumar; Gupta, Deepak Prasad; Park, Sung Hee; Kim, Jae-Hong; Lee, Sun-Hwa; Lee, In-Kyu; Sim, Taebo; Bae, Yong Chul; Lee, Won-Ha; Suk, Kyoungho |
2019-05 | Raman-Based in Situ Monitoring of Changes in Molecular Signatures during Mitochondrially Mediated Apoptosis | Shin, Hyeon Jeong; Lee, Ji Hye; Kim, Yong Duk; Shin, Injae; Sim, Taebo; Lim, Dong-Kwon |
2019-06 | Leveraging Compound Promiscuity to Identify Targetable Cysteines within the Kinome | Rao, Suman; Gurbani, Deepak; Du, Guangyan; Everley, Robert A.; Browne, Christopher M.; Chaikuad, Apirat; Tan, Li; Schroeder, Martin; Gondi, Sudershan; Ficarro, Scott B.; Sim, Taebo; Kim, Nam Doo; Berberich, Matthew J.; Knapp, Stefan; Marto, Jarrod A.; Westover, Kenneth D.; Sorger, Peter K.; Gray, Nathanael S. |
2019-06 | Discovery of Covalent CDK14 Inhibitors with Pan-TAIRE Family Specificity | Ferguson, Fleur M.; Doctor, Zainab M.; Ficarro, Scott B.; Browne, Christopher M.; Marto, Jarrod A.; Johnson, Jared L.; Yaron, Tomer M.; Cantley, Lewis C.; Kim, Nam Doo; Sim, Taebo; Berberich, Matthew J.; Kalocsay, Marian; Sorger, Peter K.; Gray, Nathanael S. |
2019-01 | Procaspase activating compound 1 controls tetracycline repressor-regulated gene expression system | Song, Chiman; Kim, Namkyoung; Park, Miri; Lee, Jiyeon; Oh, Ki-Bong; Sim, Taebo |
2019-09-26 | Identification of Novel Resorcinol Amide Derivatives as Potent and Specific Pyruvate Dehydrogenase Kinase (PDHK) Inhibitors | Cho, Hanna; Shin, Injae; Cho, Kyungseon; Yoon, Hojong; Yoo, Eun Kyung; Kim, Mi-Jin; Park, Sungmi; Lee, In-Kyu; Kim, Nam Doo; Sim, Taebo |
2019-08 | Synthesis and structure activity relationships of a series of 4-amino-1H-pyrazoles as covalent inhibitors of CDK14 | Ferguson, Fleur M.; Doctor, Zainab M.; Ficarro, Scott B.; Marto, Jarrod A.; Kim, Nam Doo; Sim, Taebo; Gray, Nathanael S. |
2019-10-24 | Identification of a Unique Resorcylic Acid Lactone Derivative That Targets Both Lymphangiogenesis and Angiogenesis | Han, Youngsun; Sengupta, Sandip; Lee, Byung Joo; Cho, Hanna; Kim, Jiknyeo; Choi, Hwan Geun; Dash, Uttam; Kim, Jin Hyoung; Kim, Nam Doo; Kim, Jeong Hun; Sim, Taebo |